Compile Data Set for Download or QSAR
maximum 50k data
Found 57 Enz. Inhib. hit(s) with all data for entry = 50013071
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50184359((3S,6S,9R,12S,15S,23S)-15-((S)-2-acetylamino-hexan...)
Affinity DataIC50:  1nMAssay Description:Binding affinity towards human melanocortin receptor (hMC1R) using NDP-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50184359((3S,6S,9R,12S,15S,23S)-15-((S)-2-acetylamino-hexan...)
Affinity DataIC50:  2nMAssay Description:Binding affinity towards human melanocortin receptor (hMC4R) using NDP-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126087(CHEMBL415341 | MT-II cyclic peptide derivative)
Affinity DataIC50:  15nMAssay Description:Binding affinity towards human melanocortin receptor (hMC1R) using NDP-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126085(CHEMBL384036 | MT-II cyclic peptide derivative)
Affinity DataIC50:  675nMAssay Description:Agonistic activity against human melanocortin receptor (hMC4R) for cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126085(CHEMBL384036 | MT-II cyclic peptide derivative)
Affinity DataIC50:  675nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126087(CHEMBL415341 | MT-II cyclic peptide derivative)
Affinity DataIC50:  5.82E+3nMAssay Description:Binding affinity towards human melanocortin receptor (hMC1R) using NDP-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126085(CHEMBL384036 | MT-II cyclic peptide derivative)
Affinity DataIC50:  1.47E+4nMAssay Description:Binding affinity towards human melanocortin receptor (hMC1R) using NDP-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126085(CHEMBL384036 | MT-II cyclic peptide derivative)
Affinity DataIC50:  1.48E+4nMAssay Description:Agonistic activity against human melanocortin receptor (hMC1R) for cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126091(CHEMBL216474 | MT-II cyclic peptide derivative)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126092(CHEMBL2371902 | MT-II cyclic peptide derivative)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126089(CHEMBL2371913 | MT-II cyclic peptide derivative)
Affinity DataEC50:  900nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126093(CHEMBL386871 | MT-II cyclic peptide derivative)
Affinity DataEC50:  480nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126094(CHEMBL437822 | MT-II cyclic peptide derivative)
Affinity DataEC50:  1.33E+3nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126095((12S,16S,23R)-15-(2-Acetylamino-hexanoylamino)-9-b...)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126092(CHEMBL2371902 | MT-II cyclic peptide derivative)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126096(CHEMBL439361 | MT-II cyclic peptide derivative)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126086(CHEMBL24892 | MT-II cyclic peptide derivative)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126097(CHEMBL264337 | MT-II cyclic peptide derivative)
Affinity DataEC50:  480nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126098(CHEMBL262437 | MT-II cyclic peptide derivative)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126099(CHEMBL410148 | MT-II cyclic peptide derivative)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126090(CHEMBL407754 | MT-II cyclic peptide derivative)
Affinity DataEC50:  65nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126096(CHEMBL439361 | MT-II cyclic peptide derivative)
Affinity DataEC50:  1.28E+3nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126088(CHEMBL409786 | MT-II cyclic peptide derivative)
Affinity DataEC50:  53nMAssay Description:Agonistic activity against human melanocortin receptor (hMC1R) for cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126094(CHEMBL437822 | MT-II cyclic peptide derivative)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126087(CHEMBL415341 | MT-II cyclic peptide derivative)
Affinity DataEC50:  4nMAssay Description:Agonistic activity against human melanocortin receptor (hMC4R) for cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126102(CHEMBL2371903 | MT-II cyclic peptide derivative)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126087(CHEMBL415341 | MT-II cyclic peptide derivative)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126086(CHEMBL24892 | MT-II cyclic peptide derivative)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126103(CHEMBL406636 | MT-II cyclic peptide derivative)
Affinity DataEC50:  176nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126104(CHEMBL2371888 | MT-II cyclic peptide derivative)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126083(CHEMBL2371887 | MT-II cyclic peptide derivative)
Affinity DataEC50:  420nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126093(CHEMBL386871 | MT-II cyclic peptide derivative)
Affinity DataEC50:  45nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126101(CHEMBL438286 | MT-II cyclic peptide derivative)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126097(CHEMBL264337 | MT-II cyclic peptide derivative)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126099(CHEMBL410148 | MT-II cyclic peptide derivative)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126105(CHEMBL2371880 | MT-II cyclic peptide derivative)
Affinity DataEC50:  735nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126084(CHEMBL412174 | MT-II cyclic peptide derivative)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126105(CHEMBL2371880 | MT-II cyclic peptide derivative)
Affinity DataEC50:  735nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126102(CHEMBL2371903 | MT-II cyclic peptide derivative)
Affinity DataEC50:  2nMAssay Description:Binding affinity towards human melanocortin receptor (hMC4R) using NDP-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50184359((3S,6S,9R,12S,15S,23S)-15-((S)-2-acetylamino-hexan...)
Affinity DataEC50:  0.600nMAssay Description:Binding affinity towards human melanocortin receptor (hMC4R) using NDP-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126088(CHEMBL409786 | MT-II cyclic peptide derivative)
Affinity DataEC50:  53nMAssay Description:Agonistic activity against human melanocortin receptor (hMC4R) for cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50184359((3S,6S,9R,12S,15S,23S)-15-((S)-2-acetylamino-hexan...)
Affinity DataEC50:  0.600nMAssay Description:Agonistic activity against human melanocortin receptor (hMC1R) for cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126102(CHEMBL2371903 | MT-II cyclic peptide derivative)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126102(CHEMBL2371903 | MT-II cyclic peptide derivative)
Affinity DataEC50:  2nMAssay Description:Agonistic activity against human melanocortin receptor (hMC4R) for cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126085(CHEMBL384036 | MT-II cyclic peptide derivative)
Affinity DataEC50:  105nMAssay Description:Agonistic activity against human melanocortin receptor (hMC1R) for cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126085(CHEMBL384036 | MT-II cyclic peptide derivative)
Affinity DataEC50:  105nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126101(CHEMBL438286 | MT-II cyclic peptide derivative)
Affinity DataEC50:  15nMAssay Description:Binding affinity towards human melanocortin receptor (hMC4R) using NDP-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126087(CHEMBL415341 | MT-II cyclic peptide derivative)
Affinity DataEC50:  4nMAssay Description:Agonistic activity against human melanocortin receptor (hMC4R) for cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126089(CHEMBL2371913 | MT-II cyclic peptide derivative)
Affinity DataEC50:  900nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126090(CHEMBL407754 | MT-II cyclic peptide derivative)
Affinity DataEC50:  370nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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