Affinity DataKi: 37nMAssay Description:Binding affinity (in vitro) against Opioid receptor delta 1 using radio-ligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.24E+3nMAssay Description:Binding affinity (in vitro) against Dopamine receptor D3 using radio-ligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.56E+3nMAssay Description:Binding affinity towards pig 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.09E+3nMAssay Description:Binding affinity (in vitro) against 5-hydroxytryptamine 1D receptor alpha using radio-ligand binding assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataIC50: 2.82E+8nMAssay Description:logIC50 (30 uM) GABA-A receptor alpha-1-beta-2-gamma-2 subunits expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataEC50: 3.60E+3nMAssay Description:Effective concentration against human recombinant GABA-A receptor alpha-1-beta-2-gamma-2 subunits expressed in Xenopus oocytesMore data for this Ligand-Target Pair