Compile Data Set for Download or QSAR
maximum 50k data
Found 123 Enz. Inhib. hit(s) with all data for entry = 50015535
LigandPNGBDBM13389(4-{[(4-cyanophenyl)methoxy](1-methyl-1H-imidazol-5...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157254(5-[(4-Cyano-benzyloxy)-(3-methyl-3H-imidazol-4-yl)...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157235(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of Farnesyl transeferase inhibitor (ABT-839)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM17325((2S)-2-[(4-{[butyl(2-cyclohexylethyl)amino]methyl}...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
LigandPNGBDBM50157238(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157256(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157270(6''-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157277(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157237(2'',3''-Dichloro-5-[(4-cyano-benzyloxy)-(3-methyl-...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157285(5-[(3,4-Dichloro-benzyloxy)-(3-methyl-3H-imidazol-...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157258(CHEMBL361353 | N-(1-{3-Cyano-6-[(6-cyano-2''-trifl...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157246(6''-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157259(5-[(4-Cyano-benzyloxy)-(3-methyl-3H-imidazol-4-yl)...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157250(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  2nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157249(5-[(4-Cyano-benzyloxy)-(3-methyl-3H-imidazol-4-yl)...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157260(2-(4-Acetyl-piperazin-1-yl)-6-[(6-cyano-2''-triflu...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157240(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157247(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157273((R)-1-{3-Cyano-6-[(6-cyano-2''-trifluoromethyl-bip...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157248(5-[(4-Cyano-benzyloxy)-(3-methyl-3H-imidazol-4-yl)...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157248(5-[(4-Cyano-benzyloxy)-(3-methyl-3H-imidazol-4-yl)...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157253(5-[(4-Fluoro-3-trifluoromethyl-benzyloxy)-(3-methy...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157257(5-[(4-Cyano-benzyloxy)-(3-methyl-3H-imidazol-4-yl)...)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157252(5-[(3-Fluoro-4-trifluoromethyl-benzyloxy)-(3-methy...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157294(4-[(6-Cyano-2''-methyl-biphenyl-3-yl)-(3-methyl-3H...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157271(2''-Methyl-5-[(3-methyl-3H-imidazol-4-yl)-(4-nitro...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157235(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157267(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157244(2''-Methyl-5-[(3-methyl-3H-imidazol-4-yl)-(3-trifl...)
Affinity DataIC50:  8.10nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157272(2''-Methyl-5-[(3-methyl-3H-imidazol-4-yl)-(3-trifl...)
Affinity DataIC50:  8.30nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157281(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  9nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157242(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157236(6-[(6-Cyano-2''-trifluoromethyl-biphenyl-3-yl)-(3-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157297(5-[(4-Chloro-benzyloxy)-(3-methyl-3H-imidazol-4-yl...)
Affinity DataIC50:  11nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157280(5-[(4-Bromo-benzyloxy)-(3-methyl-3H-imidazol-4-yl)...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157275(2''-Methyl-5-[(3-methyl-3H-imidazol-4-yl)-(4-trifl...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157245(5-[(2,6-Dichloro-pyridin-4-ylmethoxy)-(3-methyl-3H...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157263(5-[(4-Iodo-benzyloxy)-(3-methyl-3H-imidazol-4-yl)-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157293(5-[(Biphenyl-4-ylmethoxy)-(3-methyl-3H-imidazol-4-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157298(5-[(3-Bromo-benzyloxy)-(3-methyl-3H-imidazol-4-yl)...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157239(2''-Cyano-5''-[(4-cyano-benzyloxy)-(3-methyl-3H-im...)
Affinity DataIC50:  14nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157289(5-[(5,6-Dichloro-pyridin-3-ylmethoxy)-(3-methyl-3H...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157279(2''-Methyl-5-[(3-methyl-3H-imidazol-4-yl)-(4-trifl...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157278(2''-Methyl-5-[(3-methyl-3H-imidazol-4-yl)-(naphtha...)
Affinity DataIC50:  17nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM13389(4-{[(4-cyanophenyl)methoxy](1-methyl-1H-imidazol-5...)
Affinity DataIC50:  18nMAssay Description:Inhibition of Bovine Geranyl geranyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157291(5-[(3-Cyano-benzyloxy)-(3-methyl-3H-imidazol-4-yl)...)
Affinity DataIC50:  18nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157269(5-[(3,5-Dichloro-benzyloxy)-(3-methyl-3H-imidazol-...)
Affinity DataIC50:  19nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157261(5-[(3-Chloro-benzyloxy)-(3-methyl-3H-imidazol-4-yl...)
Affinity DataIC50:  19nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157264(5-[(3-Iodo-benzyloxy)-(3-methyl-3H-imidazol-4-yl)-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157268(5-[(3,4-Dichloro-benzyloxy)-(3-methyl-3H-imidazol-...)
Affinity DataIC50:  27nMAssay Description:Inhibition of Bovine farnesyl transeferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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