Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50015608
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158330((+/-)isobutyl 8-chloro-2-((4-(diethylamino)phenyl)...)
Affinity DataIC50:  2nMAssay Description:Binding affinity to GHSRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158329((+/-)-isobutyl 2-({[4-(diethylamino)phenyl]amino}c...)
Affinity DataIC50:  11nMAssay Description:Binding affinity to GHSRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158327((+/-)isobutyl 2-((4-(diethylamino)phenyl)carbamoyl...)
Affinity DataIC50:  16nMAssay Description:Binding affinity to GHSRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158327((+/-)isobutyl 2-((4-(diethylamino)phenyl)carbamoyl...)
Affinity DataIC50:  29nMAssay Description:Antagonist activity at GHSR expressed in CHOK cells assessed as inhibition of ghrelin-induced increase in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158328((+/-)-tert-butyl 2-({[4-(diethylamino)phenyl]amino...)
Affinity DataIC50:  120nMAssay Description:Binding affinity to GHSRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50153535(3-(2,6-Dichloro-phenyl)-5-methyl-isoxazole-4-carbo...)
Affinity DataIC50:  130nMAssay Description:Binding affinity to GHSRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158331((+/-)-1,2,3,4-tetrahydro-naphthalene-2-carboxylic ...)
Affinity DataIC50:  2.70E+3nMAssay Description:Binding affinity to GHSRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158327((+/-)isobutyl 2-((4-(diethylamino)phenyl)carbamoyl...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of hERG receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed