Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50016531
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50065796((E)-2-(3,4-dihydroxystyryl)-8-hydroxyquinoline-7-c...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50065796((E)-2-(3,4-dihydroxystyryl)-8-hydroxyquinoline-7-c...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170145(CHEMBL189128 | {2-[(E)-2-(3,4-Dihydroxy-phenyl)-vi...)
Affinity DataIC50:  7.00E+4nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170149((3,4-Difluoro-phenyl)-{2-[(E)-2-(3,4-dihydroxy-phe...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170144(CHEMBL188293 | {2-[(E)-2-(3,4-Dihydroxy-phenyl)-vi...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170144(CHEMBL188293 | {2-[(E)-2-(3,4-Dihydroxy-phenyl)-vi...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170148(CHEMBL188712 | {2-[(E)-2-(3,4-Dihydroxy-phenyl)-vi...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170148(CHEMBL188712 | {2-[(E)-2-(3,4-Dihydroxy-phenyl)-vi...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170145(CHEMBL189128 | {2-[(E)-2-(3,4-Dihydroxy-phenyl)-vi...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170146(CHEMBL187452 | {2-[(E)-2-(3,4-Dihydroxy-phenyl)-vi...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170146(CHEMBL187452 | {2-[(E)-2-(3,4-Dihydroxy-phenyl)-vi...)
Affinity DataIC50:  1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Unité

Curated by ChEMBL
LigandPNGBDBM50170149((3,4-Difluoro-phenyl)-{2-[(E)-2-(3,4-dihydroxy-phe...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed