Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 50018488
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196377(5-[4-(4-bromo-phenylamino)-phenylamino]-3-hydroxy-...)
Affinity DataIC50:  87nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196371(5-[4-(4-bromo-phenylamino)-phenylamino]-3-hydroxy-...)
Affinity DataIC50:  140nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196373(5-[4-(4-bromo-phenylamino)-phenylamino]-3-hydroxy-...)
Affinity DataIC50:  220nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196382(5-[4-(4-bromo-phenylamino)-phenylamino]-N-cyclohex...)
Affinity DataIC50:  300nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196374(5-[4-(4-bromo-phenylamino)-phenylamino]-3-hydroxy-...)
Affinity DataIC50:  310nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196390(3-hydroxy-N-isopropyl-5-(4-phenylamino-phenylamino...)
Affinity DataIC50:  420nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196392(3-hydroxy-N-(2-hydroxy-1-methyl-ethyl)-5-(4-phenyl...)
Affinity DataIC50:  460nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196393(5-[4-(4-bromo-phenylamino)-phenylamino]-3-hydroxy-...)
Affinity DataIC50:  460nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196383(5-[4-(4-bromo-phenylamino)-phenylamino]-N-(2,3-dih...)
Affinity DataIC50:  470nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196378(CHEMBL401105 | N-(2,3-dihydroxy-propyl)-3-hydroxy-...)
Affinity DataIC50:  900nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196369(3-hydroxy-N-(2-hydroxy-ethyl)-5-(4-phenylamino-phe...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196385(3-hydroxy-N-(4-hydroxy-butyl)-5-(4-phenylamino-phe...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196372(CHEMBL253541 | N-cyclohexylmethyl-3-hydroxy-5-(4-p...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196387(3-hydroxy-N-isopropyl-5-(4-phenoxy-phenylamino)-is...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196389(5-(4-benzoyl-phenylamino)-N-cyclohexylmethyl-3-hyd...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196370(5-(4-benzyl-phenylamino)-3-hydroxy-N-isopropyl-iso...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196388(CHEMBL399151 | N-cyclohexylmethyl-3-hydroxy-5-(4-p...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196381(3-hydroxy-N-isopropyl-5-(4-phenylazo-phenylamino)-...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196384(CHEMBL438150 | N-(2,3-dihydroxy-propyl)-3-hydroxy-...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196380(CHEMBL251629 | N-cyclohexylmethyl-3-hydroxy-5-(4-p...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196391(5-(4-cyclohexyl-phenylamino)-3-hydroxy-N-isopropyl...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196386(5-(4-benzyl-phenylamino)-N-cyclohexylmethyl-3-hydr...)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196379(5-(4-benzenesulfonyl-phenylamino)-3-hydroxy-N-isop...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196375(CHEMBL251471 | N-cyclohexylmethyl-3-hydroxy-5-(4-p...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Valeant Pharmaceutical Research And Development 3300 Hyland Avenue

Curated by ChEMBL
LigandPNGBDBM50196376(3-hydroxy-N-(2-hydroxy-1-methyl-ethyl)-5-(4-pyrazo...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of Chk2 kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed