TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of [125I]beta-CIT from rat SERT expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Yale University
Curated by ChEMBL
Yale University
Curated by ChEMBL
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of [3H]5HT uptake at rat SERT expressed in HeLa cellsMore data for this Ligand-Target Pair
Affinity DataKd: 2.82nMAssay Description:Displacement of [125I]beta-CIT from human SERT in human platelet membrane in presence of 5 uM ibogaineMore data for this Ligand-Target Pair
Affinity DataKd: 0.880nMAssay Description:Displacement of [125I]beta-CIT from human SERT in human platelet plasma membraneMore data for this Ligand-Target Pair