Compile Data Set for Download or QSAR
maximum 50k data
Found 41 Enz. Inhib. hit(s) with all data for entry = 50038160
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  3nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372555(CHEMBL272099)
Affinity DataKi:  23nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  125nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  300nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372555(CHEMBL272099)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372554(CHEMBL258295)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372554(CHEMBL258295)
Affinity DataKi:  4.20E+3nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372552(CHEMBL403722)
Affinity DataKi:  4.50E+3nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372557(CHEMBL257040)
Affinity DataKi:  6.70E+3nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372557(CHEMBL257040)
Affinity DataKi:  9.10E+3nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372552(CHEMBL403722)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372555(CHEMBL272099)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372554(CHEMBL258295)
Affinity DataKi: >2.50E+4nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372553(CHEMBL256630)
Affinity DataKi: >2.50E+4nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372552(CHEMBL403722)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372553(CHEMBL256630)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372556(CHEMBL429742)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372556(CHEMBL429742)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372556(CHEMBL429742)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372553(CHEMBL256630)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372553(CHEMBL256630)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372552(CHEMBL403722)
Affinity DataEC50: >2.50E+4nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataEC50:  5nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372554(CHEMBL258295)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at human MC4 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372557(CHEMBL257040)
Affinity DataEC50: >2.50E+4nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372556(CHEMBL429742)
Affinity DataEC50: >5.00E+4nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372553(CHEMBL256630)
Affinity DataEC50: >5.00E+4nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372553(CHEMBL256630)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372556(CHEMBL429742)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372552(CHEMBL403722)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372555(CHEMBL272099)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372555(CHEMBL272099)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372554(CHEMBL258295)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372552(CHEMBL403722)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372556(CHEMBL429742)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372557(CHEMBL257040)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372557(CHEMBL257040)
Affinity DataEC50: >1.50E+4nMAssay Description:Agonist activity at human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50372555(CHEMBL272099)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed