Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50038760
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255529(Ac-Lys(CoA)-NH2 | CHEMBL505121)
Affinity DataIC50:  980nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255522(Ac-ARTKQTARKSTGGK(CoA)APRKQL | CHEMBL526343)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255524(Ac-SGRGK(CoA)GGKGLGKGGAKRHRK | CHEMBL505605)
Affinity DataIC50:  2.88E+3nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255526(Ac-SGRGKGGKGLGK(CoA)GGAKRHRK | CHEMBL500256)
Affinity DataIC50:  4.35E+3nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255527(Ac-SGRGKGGKGLGKGGAK(CoA)RHRK | CHEMBL504265)
Affinity DataIC50:  6.62E+3nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255522(Ac-ARTKQTARKSTGGK(CoA)APRKQL | CHEMBL526343)
Affinity DataIC50:  7.54E+3nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255525(Ac-SGRGKGGK(CoA)GLGKGGAKRHRK | CHEMBL448227)
Affinity DataIC50:  8.15E+3nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50292429(2-Hydroxy-6-pentadecyl-benzoic acid | 2-Pentadecyl...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of TIP60 in human HeLa cell extracts by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255527(Ac-SGRGKGGKGLGKGGAK(CoA)RHRK | CHEMBL504265)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255528(Ac-SGRGK(CoA)QGGKARAKAKTRSSRA | CHEMBL509144)
Affinity DataIC50:  1.74E+4nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255528(Ac-SGRGK(CoA)QGGKARAKAKTRSSRA | CHEMBL509144)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255526(Ac-SGRGKGGKGLGK(CoA)GGAKRHRK | CHEMBL500256)
Affinity DataIC50:  2.59E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255529(Ac-Lys(CoA)-NH2 | CHEMBL505121)
Affinity DataIC50:  2.98E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50067040(((E,E)-1,7-bis(4-hydroxy-3-methoxyphenyl)-1,6-hept...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50367033(COENZYME_A)
Affinity DataIC50:  4.19E+4nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50367033(COENZYME_A)
Affinity DataIC50:  4.59E+4nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255526(Ac-SGRGKGGKGLGK(CoA)GGAKRHRK | CHEMBL500256)
Affinity DataIC50:  5.36E+4nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255527(Ac-SGRGKGGKGLGKGGAK(CoA)RHRK | CHEMBL504265)
Affinity DataIC50:  5.85E+4nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255528(Ac-SGRGK(CoA)QGGKARAKAKTRSSRA | CHEMBL509144)
Affinity DataIC50:  6.05E+4nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255524(Ac-SGRGK(CoA)GGKGLGKGGAKRHRK | CHEMBL505605)
Affinity DataIC50:  6.59E+4nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255522(Ac-ARTKQTARKSTGGK(CoA)APRKQL | CHEMBL526343)
Affinity DataIC50:  7.96E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50367033(COENZYME_A)
Affinity DataIC50:  8.23E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255529(Ac-Lys(CoA)-NH2 | CHEMBL505121)
Affinity DataIC50:  1.08E+5nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255525(Ac-SGRGKGGK(CoA)GLGKGGAKRHRK | CHEMBL448227)
Affinity DataIC50:  1.12E+5nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255525(Ac-SGRGKGGK(CoA)GLGKGGAKRHRK | CHEMBL448227)
Affinity DataIC50:  1.24E+5nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255524(Ac-SGRGK(CoA)GGKGLGKGGAKRHRK | CHEMBL505605)
Affinity DataIC50:  1.43E+5nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50067040(((E,E)-1,7-bis(4-hydroxy-3-methoxyphenyl)-1,6-hept...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50292429(2-Hydroxy-6-pentadecyl-benzoic acid | 2-Pentadecyl...)
Affinity DataIC50:  3.75E+5nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50292429(2-Hydroxy-6-pentadecyl-benzoic acid | 2-Pentadecyl...)
Affinity DataIC50:  6.67E+5nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50292429(2-Hydroxy-6-pentadecyl-benzoic acid | 2-Pentadecyl...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed