Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50028032
TargetPoly [ADP-ribose] polymerase 1(Bos taurus)
University Of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)
Affinity DataIC50:  240nMAssay Description:Inhibition of calf thymus PARP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255329(2-Methylquinoline-8-carboxamide | CHEMBL471966)
Affinity DataIC50:  500nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255330(2-ethylquinoline-8-carboxamide | CHEMBL526128)
Affinity DataIC50:  800nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255331(2-phenylquinoline-8-carboxamide | CHEMBL480429)
Affinity DataIC50:  900nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255383(2-(4-methoxyphenyl)quinoline-8-carboxamide | CHEMB...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255266(CHEMBL502330 | Quinoline-8-carboxamide)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255325(3-Prop-1-ynylquinoline-8-carboxamide | CHEMBL50490...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255268(3-Ethynylquinoline-8-carboxamide | CHEMBL501330)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255267(3-Methylquinoline-8-carboxamide | CHEMBL504998)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255269(3-Ethylquinoline-8-carboxamide | CHEMBL453989)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255270(3-Ethenylquinoline-8-carboxamide | CHEMBL481793)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255264(3-Phenylquinoline-8-carboxamide | CHEMBL450259)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255384(1-Oxo-3-phenylquinoline-8-carboxamide | CHEMBL4818...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255328(3-(4-cyanophenyl)quinoline-8-carboxamide | CHEMBL4...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255327(3-(4-Methylphenyl)quinoline-8-carboxamide | CHEMBL...)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255265(3-(3-(trifluoromethyl)phenyl)quinoline-8-carboxami...)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50255326(3-(4-methoxyphenyl)quinoline-8-carboxamide | CHEMB...)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of human recombinant PARP1 by Trevigen colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed