Compile Data Set for Download or QSAR
maximum 50k data
Found 56 Enz. Inhib. hit(s) with all data for entry = 50028342
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257967(CHEMBL494748 | N-(2-(7-(4-chloro-3-(trifluoromethy...)
Affinity DataIC50:  0.0500nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257758(3-(2-(4-methoxyphenyl)-3-oxo-6-(3-(trifluoromethyl...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257968(CHEMBL494359 | N-(2-(7-(4-fluoro-3-methylbenzylami...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257922(CHEMBL494544 | N-(2-(3-(4-ethylphenyl)-2-oxo-7-(3-...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257920(CHEMBL493961 | N-(2-(3-(4-methoxyphenyl)-2-oxo-7-(...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258152(3-(6-(4-methoxyphenyl)-7-oxo-2-(3-(trifluoromethyl...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258016(CHEMBL522160 | N-(2-(3-(4-methoxyphenyl)-2-oxo-7-(...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257919(CHEMBL493960 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258196(3-(7-oxo-6-p-tolyl-2-(3-(trifluoromethyl)benzylami...)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257809(CHEMBL495170 | N-(2-(6-(3-chloro-4-fluorobenzylami...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257921(CHEMBL494543 | N-(2-(2-oxo-3-(pyridin-3-yl)-7-(3-(...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257965(CHEMBL494552 | N-(2-(3-(4-methoxyphenyl)-7-(3-meth...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257808(CHEMBL495001 | N-(2-(6-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257757(3-(6-(3,4-dichlorobenzylamino)-2-(4-methoxyphenyl)...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257553(CHEMBL523668 | N-(2-(6-(4-fluoro-3-(trifluoromethy...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257861(CHEMBL495359 | N-(2-(7-(3,4-dichlorobenzylamino)-2...)
Affinity DataIC50:  21nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257967(CHEMBL494748 | N-(2-(7-(4-chloro-3-(trifluoromethy...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257919(CHEMBL493960 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257860(CHEMBL495194 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257919(CHEMBL493960 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257967(CHEMBL494748 | N-(2-(7-(4-chloro-3-(trifluoromethy...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258014(CHEMBL494750 | N-(2-(2-(3,4-dichlorobenzylamino)-6...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258197(CHEMBL495191 | N-(2-(6-(3,4-dichlorobenzylamino)-2...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257757(3-(6-(3,4-dichlorobenzylamino)-2-(4-methoxyphenyl)...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257758(3-(2-(4-methoxyphenyl)-3-oxo-6-(3-(trifluoromethyl...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257808(CHEMBL495001 | N-(2-(6-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257757(3-(6-(3,4-dichlorobenzylamino)-2-(4-methoxyphenyl)...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257758(3-(2-(4-methoxyphenyl)-3-oxo-6-(3-(trifluoromethyl...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257860(CHEMBL495194 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta6-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258197(CHEMBL495191 | N-(2-(6-(3,4-dichlorobenzylamino)-2...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258014(CHEMBL494750 | N-(2-(2-(3,4-dichlorobenzylamino)-6...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Rattus norvegicus)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257808(CHEMBL495001 | N-(2-(6-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257860(CHEMBL495194 | N-(2-(7-(3,4-dichlorobenzylamino)-3...)
Affinity DataIC50:  34nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258154(3-(2-(3,4-dichlorobenzylamino)-7-oxo-6-(pyridin-3-...)
Affinity DataIC50:  36nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257862(CHEMBL522883 | N-(2-(7-(3,4-dichlorobenzylamino)-2...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258241(CHEMBL494032 | N-(2-(2-(4-methoxyphenyl)-3-oxo-6-(...)
Affinity DataIC50:  47nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258240(CHEMBL494031 | N-(2-(6-(3-chloro-4-fluorobenzylami...)
Affinity DataIC50:  47nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257501(CHEMBL522492 | N-(2-(6-(3,5-bis(trifluoromethyl)be...)
Affinity DataIC50:  51nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258197(CHEMBL495191 | N-(2-(6-(3,4-dichlorobenzylamino)-2...)
Affinity DataIC50:  81nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258155(3-(7-oxo-6-(pyridin-3-yl)-2-(3-(trifluoromethyl)be...)
Affinity DataIC50:  92nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257700(CHEMBL493929 | N-(2-(2-(4-methoxyphenyl)-6-(3-meth...)
Affinity DataIC50:  96nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258238(CHEMBL494023 | N-(2-(6-(3-chlorobenzylamino)-2-(4-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258198(CHEMBL495356 | N-(2-(6-(4-chlorobenzylamino)-2-(4-...)
Affinity DataIC50:  110nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257759(3-(2-(4-methoxyphenyl)-3-oxo-6-(3-(trifluoromethyl...)
Affinity DataIC50:  120nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257810(CHEMBL521865 | N-(2-(3-oxo-2-(pyridin-3-yl)-6-(3-(...)
Affinity DataIC50:  120nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257966(CHEMBL494747 | N-(2-(7-(3,4-dimethylbenzylamino)-3...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258102(3-(2-(3,4-dichlorobenzylamino)-6-(4-methoxyphenyl)...)
Affinity DataIC50:  140nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257658(CHEMBL492498 | N-(2-(2-(4-methoxyphenyl)-3-oxo-6-(...)
Affinity DataIC50:  180nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50257499(CHEMBL493134 | N-(2-(2-(4-methoxyphenyl)-3-oxo-6-(...)
Affinity DataIC50:  210nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50258153(CHEMBL494827 | N-(2-(2-(3,4-dichlorobenzylamino)-7...)
Affinity DataIC50:  250nMAssay Description:Inhibition of Delta9-desaturase in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 56 total ) | Next | Last >>
Jump to: