Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50031303
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50059889((staurosporine)3-methoxy-2-methyl-4-methylamino-(2...)
Affinity DataIC50:  150nMAssay Description:Inhibition of GST-tagged MAPKAPK2 assessed as [33P] incorporation after 40 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50310786(CHEMBL1078220 | guttiferone P)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of GST-tagged MAPKAPK2 assessed as [33P] incorporation after 40 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50310785(CHEMBL1078219 | guttiferone O)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of GST-tagged MAPKAPK2 assessed as [33P] incorporation after 40 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed