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Found 8 Enz. Inhib. hit(s) with all data for entry = 50030733
TargetD-alanyl-D-alanine carboxypeptidase(Actinomadura sp. (strain R39))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50300661(3-borono-5-(2-methoxybenzamido)benzoic acid | CHEM...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of Actinomadura sp. R39 penicillin-binding protein preincubated for 60 mins before addition of substrate mixture of (R)-[2-(benzoylamino)p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanyl-D-alanine carboxypeptidase(Actinomadura sp. (strain R39))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50300664(3-borono-5-(2-phenoxyacetamido)benzoic acid | CHEM...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of Actinomadura sp. R39 penicillin-binding protein preincubated for 60 mins before addition of substrate mixture of (R)-[2-(benzoylamino)p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanyl-D-alanine carboxypeptidase(Actinomadura sp. (strain R39))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50300662(3-borono-5-(thiophene-2-carboxamido)benzoic acid |...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of Actinomadura sp. R39 penicillin-binding protein preincubated for 60 mins before addition of substrate mixture of (R)-[2-(benzoylamino)p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanyl-D-alanine carboxypeptidase(Actinomadura sp. (strain R39))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50300660(3-benzamido-5-boronobenzoic acid | CHEMBL575719)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of Actinomadura sp. R39 penicillin-binding protein preincubated for 60 mins before addition of substrate mixture of (R)-[2-(benzoylamino)p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanyl-D-alanine carboxypeptidase(Actinomadura sp. (strain R39))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50300663(3-borono-5-(2-(thiophen-2-yl)acetamido)benzoic aci...)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of Actinomadura sp. R39 penicillin-binding protein preincubated for 60 mins before addition of substrate mixture of (R)-[2-(benzoylamino)p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanyl-D-alanine carboxypeptidase(Actinomadura sp. (strain R39))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50300659(3-borono-5-(2-phenylacetamido)benzoic acid | CHEMB...)
Affinity DataIC50:  8.80E+4nMAssay Description:Inhibition of Actinomadura sp. R39 penicillin-binding protein preincubated for 60 mins before addition of substrate mixture of (R)-[2-(benzoylamino)p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-alanyl-D-alanine carboxypeptidase(Actinomadura sp. (strain R39))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50067893(3-Carboxyphenylboronicacid | 3-boronobenzoic acid ...)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of Actinomadura sp. R39 penicillin-binding protein preincubated for 60 mins before addition of substrate mixture of (R)-[2-(benzoylamino)p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPenicillin-binding protein 2x(Streptococcus pneumoniae)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50300665(5-boronothiophene-2-carboxylic acid | CHEMBL573906)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of penicillin-resistant Streptococcus pneumoniae 5204 PBP2X preincubated for 4 hrs before addition of substrate mixture of (R)-[2-(benzoyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed