Compile Data Set for Download or QSAR
maximum 50k data
Found 58 Enz. Inhib. hit(s) with all data for entry = 50030842
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302529(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(2-(4-methylp...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302531(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(pyrrolidi...)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302526(5-(3-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50:  7nMAssay Description:Inhibition of PKCepsilon by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302528(4-(4-methyl-1H-indol-5-ylamino)-5-(2-(2-(4-methylp...)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302525(5-(2-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302509(4-(4-methyl-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50:  8.30nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302532(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(2-(pyrrolidi...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302511(4-(3H-indol-4-ylamino)-5-styrylnicotinonitrile | C...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302527(5-(4-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302530(4-(4-methyl-1H-indol-5-ylamino)-5-(2-(2-(pyrrolidi...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302510(4-(1H-indol-5-ylamino)-5-styrylnicotinonitrile | C...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302531(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(pyrrolidi...)
Affinity DataIC50:  25nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302524(5-(2-cyclohexylvinyl)-4-(4-methyl-1H-indol-5-ylami...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302523(4-(4-methyl-1H-indol-5-ylamino)-5-phenethylnicotin...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302516(4-(4,7-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302528(4-(4-methyl-1H-indol-5-ylamino)-5-(2-(2-(4-methylp...)
Affinity DataIC50:  34nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302529(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(2-(4-methylp...)
Affinity DataIC50:  41nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50:  53nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302526(5-(3-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50:  62nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302518(4-(6-chloro-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50:  65nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302515(4-(2,4-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302509(4-(4-methyl-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50:  72nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302519(4-(7-chloro-4-methyl-1H-indol-5-ylamino)-5-styryln...)
Affinity DataIC50:  77nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302508((Z)-4-(4-methyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50:  79nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302532(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(2-(pyrrolidi...)
Affinity DataIC50:  81nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302521(4-(4-methyl-1H-indol-5-yloxy)-5-styrylnicotinonitr...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302511(4-(3H-indol-4-ylamino)-5-styrylnicotinonitrile | C...)
Affinity DataIC50:  96nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302525(5-(2-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50:  110nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302530(4-(4-methyl-1H-indol-5-ylamino)-5-(2-(2-(pyrrolidi...)
Affinity DataIC50:  140nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302527(5-(4-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50:  150nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302517(4-(1,4-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302510(4-(1H-indol-5-ylamino)-5-styrylnicotinonitrile | C...)
Affinity DataIC50:  240nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50:  330nMAssay Description:Inhibition of PKCeta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302508((Z)-4-(4-methyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50:  350nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302514(4-(2-methyl-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50:  360nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302524(5-(2-cyclohexylvinyl)-4-(4-methyl-1H-indol-5-ylami...)
Affinity DataIC50:  420nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302522(4-((1H-indol-5-yl)(methyl)amino)-5-styrylnicotinon...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50:  520nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50:  520nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302515(4-(2,4-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50:  620nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302523(4-(4-methyl-1H-indol-5-ylamino)-5-phenethylnicotin...)
Affinity DataIC50:  670nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302520(4-(1H-indol-5-yloxy)-5-styrylnicotinonitrile | CHE...)
Affinity DataIC50:  690nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302514(4-(2-methyl-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50:  800nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302519(4-(7-chloro-4-methyl-1H-indol-5-ylamino)-5-styryln...)
Affinity DataIC50:  880nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302518(4-(6-chloro-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of PKCbeta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302512(4-(1H-indol-6-ylamino)-5-styrylnicotinonitrile | C...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302516(4-(4,7-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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