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Found 10 Enz. Inhib. hit(s) with all data for entry = 50031663
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50316864(CHEMBL1099361 | [(2R,4S,5S)-5-(N-Boc-L-leucyl-L-ph...)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50316861(CHEMBL1099022 | N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(...)
Affinity DataIC50:  2.64E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50316860((2R,4S,5S)-4-hydroxy-N-isobutyl-2,7-dimethyl-5-((S...)
Affinity DataIC50:  3.79E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50316862(CHEMBL1099023 | N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(...)
Affinity DataIC50:  3.81E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50316863(2,4-dichloro-N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(iso...)
Affinity DataIC50:  4.24E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50316867(CHEMBL1086716 | N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(...)
Affinity DataIC50:  4.67E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50316865(CHEMBL1087609 | N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(...)
Affinity DataIC50:  6.93E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50316858(CHEMBL1088138 | N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(...)
Affinity DataIC50:  8.07E+3nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50316866(CHEMBL1087736 | N-((S)-1-((4S,5S,7R)-5-hydroxy-8-(...)
Affinity DataIC50:  1.57E+4nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50316859(CHEMBL1098682 | [(2R,4S,5S)-5-[N-(4-trifluoromethy...)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of human recombinant BACE1 using fluorescent peptide substrate after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed