Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50031178
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50308552((1'S,2'R,3'S,4'R,5'S)-4-(6-Amino-2-chloro-9H-purin...)
Affinity DataEC50:  722nMAssay Description:Activation of human P2Y1 receptor expressed in human 1321N1 cells assessed as induction of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50118242(((2R,3S,4R,5R)-5-(6-amino-2-(methylthio)-9H-purin-...)
Affinity DataEC50:  10.3nMAssay Description:Activation of human P2Y1 receptor expressed in human 1321N1 cells assessed as induction of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50308552((1'S,2'R,3'S,4'R,5'S)-4-(6-Amino-2-chloro-9H-purin...)
Affinity DataEC50:  1.89nMAssay Description:Agonist activity at human P2Y1 receptor expressed in human 1321N1 cells by PLC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed