Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50031889
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50149806(2''-Amino-6''-(2-hydroxy-phenyl)-1,2,3,4,5,6-hexah...)
Affinity DataIC50:  174nMAssay Description:Inhibition of IKKbeta by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50321061((E)-4-(4-((5-(1,3-Dioxoisoindolin-5-yl)furan-2-yl)...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of IKKbeta by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50321060((E)-N-(5-(2-(2-(4-Hydroxy-3-methoxybenzylidene)hyd...)
Affinity DataIC50:  6.98E+3nMAssay Description:Inhibition of IKKbeta by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50321059((E)-N-(5-(2-(2-(4-Hydroxy-3-methoxybenzylidene)hyd...)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of IKKbeta by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed