Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50032085
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50324078(1-(4-((4-Chlorophenyl)(phenyl)methyl)piperazin-1-y...)
Affinity DataIC50:  190nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50324082(4-(4-Isopropylbenzylamino)-1-(4-((4-chlorophenyl)(...)
Affinity DataIC50:  280nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50324076(1-(4-((4-Chlorophenyl)(phenyl)methyl)piperazin-1-y...)
Affinity DataIC50:  360nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50324075(1-(4-((4-Chlorophenyl)(phenyl)methyl)piperazin-1-y...)
Affinity DataIC50:  420nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50324080(4-(4-Nitrobenzylamino)-1-(4-((4-chlorophenyl)(phen...)
Affinity DataIC50:  600nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50117922((1S,2S)-2-(2-((3-(1H-benzo[d]imidazol-2-yl)propyl)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of T-type Cav3.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1I(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50117922((1S,2S)-2-(2-((3-(1H-benzo[d]imidazol-2-yl)propyl)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of T-type Cav3.3 channelMore data for this Ligand-Target Pair
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50117922((1S,2S)-2-(2-((3-(1H-benzo[d]imidazol-2-yl)propyl)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of T-type Cav3.1 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50324084(4-(2,6-Dichlorobenzylamino)-1-(4-((4-chlorophenyl)...)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50117922((1S,2S)-2-(2-((3-(1H-benzo[d]imidazol-2-yl)propyl)...)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50324077(4-(2-Ethylbutylamino)-1-(4-((4-chlorophenyl)(pheny...)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50324079(4-(Benzylamino)-1-(4-((4-chlorophenyl)(phenyl)meth...)
Affinity DataIC50:  1.67E+3nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50324083(4-(4-(Dimethylamino)benzylamino)-1-(4-((4-chloroph...)
Affinity DataIC50:  2.32E+3nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50324074(4-amino-1-(4-((4-chlorophenyl)(phenyl)methyl)piper...)
Affinity DataIC50:  3.71E+3nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50324081(4-(4-Methoxybenzylamino)-1-(4-((4-chlorophenyl)(ph...)
Affinity DataIC50:  1.61E+4nMAssay Description:Inhibition of T-type alpha1G channel expressed in HEK293 cells by whole-cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1I(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50017702(1-(bis(4-fluorophenyl)methyl)-4-cinnamylpiperazine...)
Affinity DataKd:  840nMAssay Description:Inhibition of T-type Cav3.3 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50019293(1-(1-{3-[Bis-(4-fluoro-phenyl)-amino]-propyl}-pipe...)
Affinity DataKd:  29nMAssay Description:Inhibition of dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50017702(1-(bis(4-fluorophenyl)methyl)-4-cinnamylpiperazine...)
Affinity DataKd:  530nMAssay Description:Inhibition of T-type Cav3.1 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetVoltage-dependent T-type calcium channel subunit alpha-1H(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50017702(1-(bis(4-fluorophenyl)methyl)-4-cinnamylpiperazine...)
Affinity DataKd:  3.60E+3nMAssay Description:Inhibition of T-type Cav3.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed