Compile Data Set for Download or QSAR
maximum 50k data
Found 118 Enz. Inhib. hit(s) with all data for entry = 50041852
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416888(CHEMBL1257363)
Affinity DataEC50:  3.63E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416889(CHEMBL1258290)
Affinity DataEC50:  2.00E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416890(CHEMBL1258291)
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416891(CHEMBL1258402)
Affinity DataEC50:  1.32E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416892(CHEMBL1258403)
Affinity DataEC50:  759nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416893(CHEMBL1258510)
Affinity DataEC50:  2.19E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416894(CHEMBL1258511)
Affinity DataEC50:  562nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416895(CHEMBL1258628)
Affinity DataEC50:  3.24E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416896(CHEMBL1258629)
Affinity DataEC50:  191nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416897(CHEMBL1258737)
Affinity DataEC50:  398nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416898(CHEMBL1258738)
Affinity DataEC50:  1.95E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416899(CHEMBL1258857)
Affinity DataEC50:  2.09E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416900(CHEMBL1258858)
Affinity DataEC50:  871nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416901(CHEMBL1258972)
Affinity DataEC50:  2.24E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416902(CHEMBL1258973)
Affinity DataEC50:  832nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416903(CHEMBL1257240)
Affinity DataEC50:  1.02E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416904(CHEMBL1257241)
Affinity DataEC50:  1.95E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416905(CHEMBL1257362)
Affinity DataEC50:  7.41E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416906(CHEMBL1257471)
Affinity DataEC50:  813nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416907(CHEMBL1257472)
Affinity DataEC50:  4.37E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416908(CHEMBL1257593)
Affinity DataEC50:  1.23E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416909(CHEMBL1257594)
Affinity DataEC50:  7.76E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416910(CHEMBL1257712)
Affinity DataEC50:  2.34E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416911(CHEMBL1257713)
Affinity DataEC50:  5.75E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416912(CHEMBL1257835)
Affinity DataEC50:  309nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416913(CHEMBL1257836)
Affinity DataEC50:  813nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416914(CHEMBL1257950)
Affinity DataEC50:  457nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416915(CHEMBL1257951)
Affinity DataEC50:  5.25E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416916(CHEMBL1258062)
Affinity DataEC50:  3.31E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416917(CHEMBL1258063)
Affinity DataEC50:  646nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416918(CHEMBL1258179)
Affinity DataEC50:  3.89E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416919(CHEMBL1258180)
Affinity DataEC50:  1.86E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416920(CHEMBL1255601)
Affinity DataEC50:  3.98E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416921(CHEMBL1258292)
Affinity DataEC50:  6.76E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416922(CHEMBL1258293)
Affinity DataEC50:  1.38E+4nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416923(CHEMBL1258404)
Affinity DataEC50:  2.75E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416924(CHEMBL1258405)
Affinity DataEC50:  3.47E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416925(CHEMBL1258512)
Affinity DataEC50:  331nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416926(CHEMBL1258513)
Affinity DataEC50:  1.51E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416927(CHEMBL1258630)
Affinity DataEC50:  1.23E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416928(CHEMBL1258631)
Affinity DataEC50:  2.09E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416929(CHEMBL1258739)
Affinity DataEC50:  1.26E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416930(CHEMBL1258740)
Affinity DataEC50:  955nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416931(CHEMBL1258859)
Affinity DataEC50:  490nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416932(CHEMBL1258860)
Affinity DataEC50:  6.03E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416933(CHEMBL1258974)
Affinity DataEC50:  1.95E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416934(CHEMBL1258975)
Affinity DataEC50:  1.58E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416935(CHEMBL1257242)
Affinity DataEC50:  676nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416936(CHEMBL1257243)
Affinity DataEC50:  813nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50416937(CHEMBL1257364)
Affinity DataEC50:  2.82E+3nMAssay Description:Inhibition of rat mGluR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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