Affinity DataKi: 3.15E+3nMAssay Description:Displacement of [3H]AMPA from recombinant GluA2 S1S2J soluble ligand binding domainMore data for this Ligand-Target Pair
Affinity DataKi: 6.87E+3nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA1 flop isoform receptor expressed in Sf9 insect cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.04E+4nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA4 flop isoform receptor expressed in Sf9 insect cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.27E+4nMAssay Description:Displacement of [3H]AMPA from recombinant rat GluA3 flop isoform receptor expressed in Sf9 insect cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at recombinant rat GluA3 flip isoform receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced cu...More data for this Ligand-Target Pair