Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50042845
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50395822(CHEMBL1762817)
Affinity DataKi:  2nMAssay Description:Binding affinity to CRF1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432097(CHEMBL2349560)
Affinity DataIC50:  0.460nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432099(CHEMBL2349558)
Affinity DataIC50:  0.460nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432098(CHEMBL2349559)
Affinity DataIC50:  0.600nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432102(CHEMBL2349570)
Affinity DataIC50:  0.610nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432103(CHEMBL2349569)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432105(CHEMBL2349567)
Affinity DataIC50:  3.20nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432108(CHEMBL2349564)
Affinity DataIC50:  4.5nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432101(CHEMBL2349571)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432106(CHEMBL2349566)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432107(CHEMBL2349565)
Affinity DataIC50:  7.40nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432111(CHEMBL2349561)
Affinity DataIC50:  7.70nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432109(CHEMBL2349563)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432110(CHEMBL2349562)
Affinity DataIC50:  19nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432100(CHEMBL2349572)
Affinity DataIC50:  53nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50432104(CHEMBL2349568)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex homogenate after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed