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Found 5 Enz. Inhib. hit(s) with all data for entry = 50043013
TargetHistone deacetylase 3(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human recombinant HDAC3 expressed in High5 insect cells using Ac-Lys-Tyr-Lys(-acetyl)-AMC as substrate after 24 hrs by fluorescence ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistone deacetylase 3(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50434531(CHEMBL2385954)
Affinity DataIC50:  830nMAssay Description:Inhibition of human recombinant HDAC3 expressed in High5 insect cells using Ac-Lys-Tyr-Lys(-acetyl)-AMC as substrate after 24 hrs by fluorescence ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50434530(CHEMBL2385955)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of human recombinant HDAC3 expressed in High5 insect cells using Ac-Lys-Tyr-Lys(-acetyl)-AMC as substrate after 24 hrs by fluorescence ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50434533(CHEMBL2385957)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of human recombinant HDAC3 expressed in High5 insect cells using Ac-Lys-Tyr-Lys(-acetyl)-AMC as substrate after 24 hrs by fluorescence ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50434532(CHEMBL2385958)
Affinity DataIC50:  8.36E+3nMAssay Description:Inhibition of human recombinant HDAC3 expressed in High5 insect cells using Ac-Lys-Tyr-Lys(-acetyl)-AMC as substrate after 24 hrs by fluorescence ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed