Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50043279
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438603(CHEMBL2414044)
Affinity DataIC50:  120nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438601(CHEMBL2414046)
Affinity DataIC50:  160nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438605(CHEMBL2414042)
Affinity DataIC50:  170nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438600(CHEMBL2414048)
Affinity DataIC50:  230nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Bos taurus)
University Of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)
Affinity DataIC50:  250nMAssay Description:Inhibition of calf thymus PARP-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438600(CHEMBL2414048)
Affinity DataIC50:  260nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)
Affinity DataIC50:  300nMAssay Description:Inhibition of PARP-1 (unknown origin) in broken nuclear preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438608(CHEMBL2414049)
Affinity DataIC50:  320nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438605(CHEMBL2414042)
Affinity DataIC50:  330nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438604(CHEMBL2414043)
Affinity DataIC50:  480nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438599(CHEMBL2414051)
Affinity DataIC50:  490nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438601(CHEMBL2414046)
Affinity DataIC50:  570nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438602(CHEMBL2414045)
Affinity DataIC50:  730nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438599(CHEMBL2414051)
Affinity DataIC50:  830nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438603(CHEMBL2414044)
Affinity DataIC50:  880nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438602(CHEMBL2414045)
Affinity DataIC50:  900nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438604(CHEMBL2414043)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438606(CHEMBL2414052)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438607(CHEMBL2414050)
Affinity DataIC50:  5.14E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50438609(CHEMBL2414047)
Affinity DataIC50:  5.61E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed