Affinity DataIC50: 110nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 148nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+3nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 1.38E+3nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 1.52E+3nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 1.67E+3nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.73E+3nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.81E+3nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
Affinity DataIC50: 1.97E+3nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 4.82E+3nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 6.35E+3nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 8.82E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.13E+4nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.63E+4nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
Affinity DataIC50: 3.13E+4nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair