Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50043714
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445015(CHEMBL3098247)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445014(CHEMBL3098249)
Affinity DataIC50:  148nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445023(CHEMBL3098234)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445011(CHEMBL3098241)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445023(CHEMBL3098234)
Affinity DataIC50:  280nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445011(CHEMBL3098241)
Affinity DataIC50:  290nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445015(CHEMBL3098247)
Affinity DataIC50:  330nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445017(CHEMBL3098242)
Affinity DataIC50:  350nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445013(CHEMBL3098250)
Affinity DataIC50:  410nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445017(CHEMBL3098242)
Affinity DataIC50:  480nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50397205(AR-C126532XX | AZD-6140 | AZD6140 | BRILINTA | TIC...)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445020(CHEMBL3098238)
Affinity DataIC50:  650nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445016(CHEMBL3098246)
Affinity DataIC50:  850nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445018(CHEMBL3098240)
Affinity DataIC50:  1.25E+3nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445019(CHEMBL3098239)
Affinity DataIC50:  1.38E+3nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445021(CHEMBL3098236)
Affinity DataIC50:  1.52E+3nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445025(CHEMBL3098243)
Affinity DataIC50:  1.67E+3nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445018(CHEMBL3098240)
Affinity DataIC50:  1.73E+3nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445022(CHEMBL3098235)
Affinity DataIC50:  1.81E+3nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445016(CHEMBL3098246)
Affinity DataIC50:  1.97E+3nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445013(CHEMBL3098250)
Affinity DataIC50:  4.82E+3nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445024(CHEMBL3098244)
Affinity DataIC50:  6.35E+3nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445011(CHEMBL3098241)
Affinity DataIC50:  8.82E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445019(CHEMBL3098239)
Affinity DataIC50:  1.13E+4nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445020(CHEMBL3098238)
Affinity DataIC50:  1.63E+4nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445012(CHEMBL3098251)
Affinity DataIC50:  3.13E+4nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed