Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50043979
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM92625(Dimethoxyquinoline, 2)
Affinity DataIC50:  100nMAssay Description:Inhibition of Syk (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50449315(CHEMBL3125863)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50449315(CHEMBL3125863)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of ZAP70 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50449314(CHEMBL3125862)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of ZAP70 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50449314(CHEMBL3125862)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50449315(CHEMBL3125863)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibition of Syk (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50449314(CHEMBL3125862)
Affinity DataIC50:  2.26E+4nMAssay Description:Inhibition of Syk (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50449314(CHEMBL3125862)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of FAK (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50449315(CHEMBL3125863)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of FAK (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50449314(CHEMBL3125862)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of c-MET (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50449315(CHEMBL3125863)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of c-MET (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed