TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataKi: 0.0520nMAssay Description:Agonist activity at alpha4beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataKi: 148nMAssay Description:Agonist activity at alpha7 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 9.5nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of human alpha4beta2 nAChR expressed in Xenopus oocytes by voltage clamp methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 106nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 132nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 152nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 153nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 338nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair