Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50042447
TargetCytochrome P450 2C11(Rattus norvegicus)
Division Of Medicinal & Process Chemistry, Division Of Parasitology, Division Of Pharmacokinetics And Metabolism, And Sophisticated Analytical Instrument Facility, Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50426305(ARTEMOTIL)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2C11 in rat liver microsome using diclofenac as substrate by HPLC-PDA analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D4(Rattus norvegicus)
Division Of Medicinal & Process Chemistry, Division Of Parasitology, Division Of Pharmacokinetics And Metabolism, And Sophisticated Analytical Instrument Facility, Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50426305(ARTEMOTIL)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2D4 in rat liver microsome using dextromethorphan as substrate by HPLC-PDA analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Rattus norvegicus)
Division Of Medicinal & Process Chemistry, Division Of Parasitology, Division Of Pharmacokinetics And Metabolism, And Sophisticated Analytical Instrument Facility, Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50426305(ARTEMOTIL)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP1A2 in rat liver microsome using phenacetin as substrate by HPLC-PDA analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed