Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50045253
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053235(CHEMBL3330232)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053242(CHEMBL3330227)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053243(CHEMBL3330148)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053238(CHEMBL3330230)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053259(CHEMBL3330133)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053234(CHEMBL3330233)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053239(CHEMBL3330229)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053231(CHEMBL3330236)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50389803(AZD7762 | CHEMBL2041933)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053233(CHEMBL3330234)
Affinity DataIC50:  9.80nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053257(CHEMBL3330135)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053256(CHEMBL3330136)
Affinity DataIC50:  14nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053236(CHEMBL3330231)
Affinity DataIC50:  15nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053260(CHEMBL3330132)
Affinity DataIC50:  16nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053232(CHEMBL3330235)
Affinity DataIC50:  23nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053230(CHEMBL3330237)
Affinity DataIC50:  25nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053241(CHEMBL3330228)
Affinity DataIC50:  41nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053258(CHEMBL3330134)
Affinity DataIC50:  48nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053254(CHEMBL3330138)
Affinity DataIC50:  116nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053251(CHEMBL3330141)
Affinity DataIC50:  178nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053231(CHEMBL3330236)
Affinity DataIC50:  202nMAssay Description:Inhibition of Aurora A (unknown origin) expressed in Escherichia coli by ZLYTETM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053235(CHEMBL3330232)
Affinity DataIC50:  328nMAssay Description:Inhibition of Aurora A (unknown origin) expressed in Escherichia coli by ZLYTETM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053259(CHEMBL3330133)
Affinity DataIC50:  495nMAssay Description:Inhibition of Aurora A (unknown origin) expressed in Escherichia coli by ZLYTETM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053260(CHEMBL3330132)
Affinity DataIC50:  791nMAssay Description:Inhibition of Aurora A (unknown origin) expressed in Escherichia coli by ZLYTETM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053243(CHEMBL3330148)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of Aurora A (unknown origin) expressed in Escherichia coli by ZLYTETM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053234(CHEMBL3330233)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of Aurora A (unknown origin) expressed in Escherichia coli by ZLYTETM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053238(CHEMBL3330230)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of Aurora A (unknown origin) expressed in Escherichia coli by ZLYTETM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053252(CHEMBL3330140)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053249(CHEMBL3330142)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053248(CHEMBL3330143)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053247(CHEMBL3330144)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053255(CHEMBL3330137)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053246(CHEMBL3330145)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053239(CHEMBL3330229)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Aurora A (unknown origin) expressed in Escherichia coli by ZLYTETM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053245(CHEMBL3330146)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053244(CHEMBL3330147)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053253(CHEMBL3330139)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Chk1 (unknown origin) by luminescent ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50053256(CHEMBL3330136)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Aurora A (unknown origin) expressed in Escherichia coli by ZLYTETM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed