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Found 8 Enz. Inhib. hit(s) with all data for entry = 50045387
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  38nMAssay Description:Inhibition of BRAF (unknown origin) incubated for 15 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human recombinant VEGFR2 incubated for 1 hr using [gamma-32P]ATP by top count assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50059791(CHEMBL3393897)
Affinity DataIC50:  531nMAssay Description:Inhibition of BRAF (unknown origin) incubated for 15 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50059790(CHEMBL3393803)
Affinity DataIC50:  650nMAssay Description:Inhibition of human recombinant VEGFR2 incubated for 1 hr using [gamma-32P]ATP by top count assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50059793(CHEMBL3393796)
Affinity DataIC50:  2.47E+3nMAssay Description:Inhibition of BRAF (unknown origin) incubated for 15 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50059790(CHEMBL3393803)
Affinity DataIC50:  1.86E+4nMAssay Description:Inhibition of human recombinant VEGFR2 incubated for 1 hr using [gamma-32P]ATP by top count assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50059791(CHEMBL3393897)
Affinity DataIC50:  2.34E+4nMAssay Description:Inhibition of human recombinant VEGFR2 incubated for 1 hr using [gamma-32P]ATP by top count assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50101400(CHEMBL3393800)
Affinity DataIC50:  4.04E+4nMAssay Description:Inhibition of human recombinant VEGFR2 incubated for 1 hr using [gamma-32P]ATP by top count assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed