Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranes incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranes incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranes incubated for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 96nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranes incubated for 15 minsMore data for this Ligand-Target Pair
Affinity DataKi: 297nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 337nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 947nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for ...More data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 95nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.800nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: >400nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for ...More data for this Ligand-Target Pair
Affinity DataEC50: 4.40nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 91nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for ...More data for this Ligand-Target Pair
Affinity DataEC50: 83nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 5.40nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair