Compile Data Set for Download or QSAR
maximum 50k data
Found 49 Enz. Inhib. hit(s) with all data for entry = 50045733
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078762(CHEMBL3416121)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078767(CHEMBL3416126)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078763(CHEMBL3416122)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078769(CHEMBL3416128)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078763(CHEMBL3416122)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078770(CHEMBL3416129)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078767(CHEMBL3416126)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078767(CHEMBL3416126)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078762(CHEMBL3416121)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078770(CHEMBL3416129)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078769(CHEMBL3416128)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078765(CHEMBL3416124)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078766(CHEMBL3416125)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078766(CHEMBL3416125)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078770(CHEMBL3416129)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078762(CHEMBL3416121)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078765(CHEMBL3416124)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078769(CHEMBL3416128)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078765(CHEMBL3416124)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranes incubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078765(CHEMBL3416124)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078765(CHEMBL3416124)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranes incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078766(CHEMBL3416125)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078763(CHEMBL3416122)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078765(CHEMBL3416124)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranes incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078765(CHEMBL3416124)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranes incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078772(CHEMBL3416120)
Affinity DataKi:  297nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078772(CHEMBL3416120)
Affinity DataKi:  337nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078772(CHEMBL3416120)
Affinity DataKi:  947nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078764(CHEMBL3416123)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078771(CHEMBL3416119)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078768(CHEMBL3416127)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078764(CHEMBL3416123)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078771(CHEMBL3416119)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078768(CHEMBL3416127)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078764(CHEMBL3416123)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078771(CHEMBL3416119)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078768(CHEMBL3416127)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078762(CHEMBL3416121)
Affinity DataEC50:  16nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50432728(CHEMBL2348461)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078770(CHEMBL3416129)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078763(CHEMBL3416122)
Affinity DataEC50:  95nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078769(CHEMBL3416128)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078769(CHEMBL3416128)
Affinity DataEC50: >400nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078766(CHEMBL3416125)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078765(CHEMBL3416124)
Affinity DataEC50:  12nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078763(CHEMBL3416122)
Affinity DataEC50:  91nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078767(CHEMBL3416126)
Affinity DataEC50:  83nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078762(CHEMBL3416121)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078767(CHEMBL3416126)
Affinity DataEC50:  5.40nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed