TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human ERG expressed in CHO cells assessed as whole cell current by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 932nMAssay Description:Inhibition of human recombinant CYP3A4 using midazolam as substrate after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.54E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using testosterone as substrate after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.74E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using testosterone as substrate after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using midazolam as substrate after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 8.11E+3nMAssay Description:Inhibition of human recombinant CYP2C19 after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 8.54E+3nMAssay Description:Inhibition of human recombinant CYP2C9 after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of human recombinant CYP2C19 after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells assessed as whole cell current by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant CYP1A2 after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant CYP2C9 after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant CYP2D6 after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant CYP2D6 after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant CYP1A2 after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair