Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50046099
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094876(CHEMBL3589129)
Affinity DataIC50:  700nMAssay Description:Inhibition of human GOAT octanoylation activity expressed in insect Sf9 cell membranes using GSSFLCAcDan as substrate after 1 hr by reverse phase HPL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094875(CHEMBL3589130)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human GOAT octanoylation activity expressed in insect Sf9 cell membranes using GSSFLCAcDan as substrate after 1 hr by reverse phase HPL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094874(CHEMBL3589131)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of human GOAT octanoylation activity expressed in insect Sf9 cell membranes using GSSFLCAcDan as substrate after 1 hr by reverse phase HPL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094877(CHEMBL3589128)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human GOAT octanoylation activity expressed in insect Sf9 cell membranes using GSSFLCAcDan as substrate after 1 hr by reverse phase HPL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed