Affinity DataKi: 0.480nMAssay Description:Displacement of [3H]-spiperone from dopamine D3 receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid scintill...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid scintill...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]-SCH-23390 from dopamine D1 receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid scintill...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-HT1A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid scintillation...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Binding affinity to 5-HT2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Binding affinity to 5-HT2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 109nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 149nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 184nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 235nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 268nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 383nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 496nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 571nMAssay Description:Displacement of [3H]-spiperone from dopamine D3 receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid scintill...More data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 1.14E+3nMAssay Description:Displacement of [3H]-spiperone from dopamine D3 receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid scintill...More data for this Ligand-Target Pair
Affinity DataKi: 1.36E+3nMAssay Description:Displacement of [3H]ketanserin hydrochloride from 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid...More data for this Ligand-Target Pair
Affinity DataKi: 1.44E+3nMAssay Description:Displacement of [3H]-spiperone from dopamine D3 receptor (unknown origin) expressed in HEK293 cell membranes incubated for 15 mins by liquid scintill...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity against 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes assessed as reduction in [35S]-GTPgammaS binding incu...More data for this Ligand-Target Pair
Affinity DataIC50: 1.37E+3nMAssay Description:Antagonist activity against 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes assessed as reduction in [35S]-GTPgammaS binding incu...More data for this Ligand-Target Pair
Affinity DataIC50: 1.66E+3nMAssay Description:Antagonist activity against 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes assessed as reduction in [35S]-GTPgammaS binding incu...More data for this Ligand-Target Pair
Affinity DataIC50: 7.43E+3nMAssay Description:Antagonist activity against 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes assessed as reduction in [35S]-GTPgammaS binding incu...More data for this Ligand-Target Pair
Affinity DataIC50: 9.12E+3nMAssay Description:Antagonist activity against 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes assessed as reduction in [35S]-GTPgammaS binding incu...More data for this Ligand-Target Pair
Affinity DataIC50: 2.13E+4nMAssay Description:Antagonist activity against 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes assessed as reduction in [35S]-GTPgammaS binding incu...More data for this Ligand-Target Pair
Affinity DataIC50: 2.77E+4nMAssay Description:Antagonist activity against 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes assessed as reduction in [35S]-GTPgammaS binding incu...More data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Agonist activity at 5-HT2A receptor (unknown origin) expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding incubated fo...More data for this Ligand-Target Pair