TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 155nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 602nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 711nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 726nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 931nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 2.33E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 8.74E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 1.59E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Alexandru Ioan Cuza University
Curated by ChEMBL
Alexandru Ioan Cuza University
Curated by ChEMBL
Affinity DataIC50: 1.93E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair