Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50010011
TargetHeat shock protein 90, putative(Plasmodium falciparum 3D7)
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Curated by ChEMBL
LigandPNGBDBM50008059(CHEBI:5292 | GELDANAMYCIN)
Affinity DataKd:  169nMAssay Description:Binding affinity to recombinant Plasmodium falciparum Hsp90 expressed in Escherichia coli BL21(DE3) pLysS by microscale thermophoresis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50008059(CHEBI:5292 | GELDANAMYCIN)
Affinity DataKd:  158nMAssay Description:Binding affinity to recombinant human Hsp90 beta expressed in Escherichia coli BL21(DE3) pLysS by microscale thermophoresis assayMore data for this Ligand-Target Pair
TargetHeat shock protein 90, putative(Plasmodium falciparum 3D7)
Universit£

Curated by ChEMBL
LigandPNGBDBM50406805(CHEMBL585793 | GNF-Pf-4574)
Affinity DataKd:  2.81E+4nMAssay Description:Binding affinity to recombinant Plasmodium falciparum Hsp90 expressed in Escherichia coli BL21(DE3) pLysS by microscale thermophoresis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein 90, putative(Plasmodium falciparum 3D7)
Universit£

Curated by ChEMBL
LigandPNGBDBM50534392(CHEMBL4446324)
Affinity DataKd:  2.56E+4nMAssay Description:Binding affinity to recombinant Plasmodium falciparum Hsp90 expressed in Escherichia coli BL21(DE3) pLysS by microscale thermophoresis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed