Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50047782
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50189885(Rohitukine)
Affinity DataIC50:  300nMAssay Description:Inhibition of human Cdk9/T1 using YSPTSPSYSPTSPSYSPTSPKKK peptide as substrate after 30 mins by 33P-ATP filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50189885(Rohitukine)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of human Cdk2/cyclin A using histone H1 substrate after 30 mins by 33P-ATP filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed