TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of GST-tagged c-Met (unknown origin) assessed as phosphotyrosine levels preincubated foe 15 mins followed by addition of poly(glutamic aci...More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of GST-tagged c-Met (unknown origin) assessed as phosphotyrosine levels preincubated foe 15 mins followed by addition of poly(glutamic aci...More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of GST-tagged c-Met (unknown origin) assessed as phosphotyrosine levels preincubated foe 15 mins followed by addition of poly(glutamic aci...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human CDK2/cyclinA expressed in Baculovirus infected T.ni cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human CDK2/cyclinA expressed in Baculovirus infected T.ni cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human CDK2/cyclinA expressed in Baculovirus infected T.ni cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 1(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human CDK1/cyclinA expressed in Baculovirus infected Sf9 cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH2...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human CDK2/cyclinA expressed in Baculovirus infected T.ni cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human CDK2/cyclinA expressed in Baculovirus infected T.ni cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human CDK2/cyclinA expressed in Baculovirus infected T.ni cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH...More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of GST-tagged c-Met (unknown origin) assessed as phosphotyrosine levels preincubated foe 15 mins followed by addition of poly(glutamic aci...More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of GST-tagged c-Met (unknown origin) assessed as phosphotyrosine levels preincubated foe 15 mins followed by addition of poly(glutamic aci...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 1(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human CDK1/cyclinA expressed in Baculovirus infected Sf9 cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH2...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 1(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of human CDK1/cyclinA expressed in Baculovirus infected Sf9 cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH2...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of human CDK2/cyclinA expressed in Baculovirus infected T.ni cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 1(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of human CDK1/cyclinA expressed in Baculovirus infected Sf9 cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH2...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 1(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of human CDK1/cyclinA expressed in Baculovirus infected Sf9 cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH2...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of human CDK2/cyclinA expressed in Baculovirus infected T.ni cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 1(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of human CDK1/cyclinA expressed in Baculovirus infected Sf9 cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH2...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 1(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of human CDK1/cyclinA expressed in Baculovirus infected Sf9 cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH2...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 1(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of human CDK1/cyclinA expressed in Baculovirus infected Sf9 cells using Biotin-aminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH2...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of GST-tagged Shp2 PTP domain (unknown origin) using DiFMUP as substrate measured after 5 to 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 4.99E+3nMAssay Description:Inhibition of human GST-tagged Shp2 (205 to 593 residues) expressed Escherichia coli DH5alpha assessed as inhibition of PTP activity using DiFMUP as ...More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 7.63E+3nMAssay Description:Inhibition of GST-tagged c-Met (unknown origin) assessed as phosphotyrosine levels preincubated foe 15 mins followed by addition of poly(glutamic aci...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of GSK-3beta (unknown origin) assessed as inhibition of phosphorylation using Ser/Thr 9 peptide as substrate by FRET-based Z-LYTE assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of GST-tagged c-Met (unknown origin) assessed as phosphotyrosine levels preincubated foe 15 mins followed by addition of poly(glutamic aci...More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of GST-tagged c-Met (unknown origin) assessed as phosphotyrosine levels preincubated foe 15 mins followed by addition of poly(glutamic aci...More data for this Ligand-Target Pair