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Found 33 Enz. Inhib. hit(s) with all data for entry = 50048062
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198338(CHEMBL3938038)
Affinity DataKi:  0.389nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200566(CHEMBL3902626)
Affinity DataKi:  0.603nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201790(CHEMBL3917716)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200441(CHEMBL3930616)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50393116(CHEMBL2153423)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201791(CHEMBL3920110)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201789(CHEMBL3946843)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200441(CHEMBL3930616)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201790(CHEMBL3917716)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198338(CHEMBL3938038)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201791(CHEMBL3920110)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200566(CHEMBL3902626)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197059(CHEMBL3976144)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197548(CHEMBL3947302)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201789(CHEMBL3946843)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197548(CHEMBL3947302)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197059(CHEMBL3976144)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50393116(CHEMBL2153423)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198439(CHEMBL3967641)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198439(CHEMBL3967641)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50393116(CHEMBL2153423)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201790(CHEMBL3917716)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201791(CHEMBL3920110)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200441(CHEMBL3930616)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198338(CHEMBL3938038)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201789(CHEMBL3946843)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197059(CHEMBL3976144)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200566(CHEMBL3902626)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201787(CHEMBL27021)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197548(CHEMBL3947302)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201787(CHEMBL27021)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198439(CHEMBL3967641)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201787(CHEMBL27021)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed