Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50012594
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Mannheim University Of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50558639(CHEMBL4789649)
Affinity DataEC50:  4.59E+4nMAssay Description:Activation of rat TRPV1 transfected in HEK293 cells assessed as increase in calcium influx in presence of capsaicin by FURA-2-AM dye based fluorescen...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Mannheim University Of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460759(CHEMBL4226014)
Affinity DataEC50:  7.10E+3nMAssay Description:Activation of rat TRPV1 transfected in HEK293 cells assessed as increase in calcium influx in presence of capsaicin by FURA-2-AM dye based fluorescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed