Affinity DataIC50: 7nMAssay Description:Inhibition of GST-tagged EED (unknown origin) after 1 hr by OG(488) as probe-based TR-FRET analysisMore data for this Ligand-Target Pair
TargetLethal(3)malignant brain tumor-like protein 1(Homo sapiens)
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataIC50: 98nMAssay Description:Inhibition of L3MBTL1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
TargetLethal(3)malignant brain tumor-like protein 1(Homo sapiens)
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataIC50: 282nMAssay Description:Inhibition of L3MBTL1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase 2A(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of recombinant SUMO-tagged MLL1 (unknown origin) by histone methyl transferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of full length N-terminal His-tagged EED (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells after 30 mins by 3-FAM labelled fluor...More data for this Ligand-Target Pair
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of full length N-terminal His-tagged EED (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells after 30 mins by 3-FAM labelled fluor...More data for this Ligand-Target Pair
Affinity DataIC50: 3.87E+3nMAssay Description:Inhibition of full length N-terminal His-tagged EED (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells after 30 mins by 3-FAM labelled fluor...More data for this Ligand-Target Pair
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of Cbx7 (unknown origin) using FITC-labeled SETDB1-K1170me3 peptide as probe by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of JARID1A PHD finger domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of N terminally fluorescein-tagged H3K27me3 binding to N terminallyHis6-tagged human Cbx7 expressed in Escherichia coli BL21 (DE3) by fluo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of 53BP1 methyllysine binding domain (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of 53BP1 methyllysine binding domain (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+4nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptor in the rabbit heartMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of recombinant HQ5-Halo-tagged JARID1A PHD3 finger domain (unknown origin) expressed in BL21(DE3)pLysS cells after 1 hr by chemiluminescen...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of recombinant HQ5-Halo-tagged JARID1A PHD3 finger domain (unknown origin) expressed in BL21(DE3)pLysS cells after 1 hr by chemiluminescen...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Competitive displacement of p53K382me2 from His-tagged 53BP1 tandem Tudor domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of Cbx7 (unknown origin) using FITC-labeled SETDB1-K1170me3 peptide as probe by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataKd: 800nMAssay Description:Inhibition of JARID1A (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 640nMAssay Description:Binding affinity to C-terminal His-tagged CDYL2 (1 to 75 residues) (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells by ITC methodMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataKd: 7.00E+3nMAssay Description:Binding affinity to GLP (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataKd: 5.00E+3nMAssay Description:Binding affinity to GLP (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 680nMAssay Description:Binding affinity to full length N-terminal His-tagged EED (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells by ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 8.80E+3nMAssay Description:Binding affinity to full length N-terminal His-tagged EED (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells by ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 4.80E+3nMAssay Description:Binding affinity to full length N-terminal His-tagged EED (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells by ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 82nMAssay Description:Binding affinity to EED (unknown origin) by ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding affinity to 15N-labeled GST-tagged ING2 PHD finger domain (212 to 264 residues) (unknown origin) expressed in Escherichia coli Rosetta2 BL21(...More data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Binding affinity to 15N-labeled GST-tagged ING2 PHD finger domain (212 to 264 residues) (unknown origin) expressed in Escherichia coli Rosetta2 BL21(...More data for this Ligand-Target Pair
Affinity DataKd: 2.90E+4nMAssay Description:Binding affinity to Cbx7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 1.09E+3nMAssay Description:Binding affinity to full length N-terminal His-tagged EED (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells by ITC methodMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataKd: 6.00E+3nMAssay Description:Binding affinity to G9a (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.20E+4nMAssay Description:Binding affinity to 53BP1 methyllysine binding domain (unknown origin) by ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 97nMAssay Description:Binding affinity to Cbx7 (unknown origin) by ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 490nMAssay Description:Binding affinity to N-terminal GST-tagged CDYL (1 to 78 residues) (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells after 30 mins by fluore...More data for this Ligand-Target Pair
Affinity DataKd: 50nMAssay Description:Binding affinity to 15N-labeled GST-tagged ING2 PHD finger domain (212 to 264 residues) (unknown origin) expressed in Escherichia coli Rosetta2 BL21(...More data for this Ligand-Target Pair
Affinity DataKd: 1.14E+3nMAssay Description:Binding affinity to full length N-terminal His-tagged EED (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells by ITC methodMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataKd: 800nMAssay Description:Inhibition of JARID1A (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase 2A(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Binding affinity to 15N-labeled GST-tagged MLL1 PHD3 finger domain (1565 to 1627 residues) (unknown origin) expressed in Escherichia coli Rosetta2 BL...More data for this Ligand-Target Pair
Affinity DataKd: 6.70E+3nMAssay Description:Binding affinity to Cbx7 (unknown origin) by ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 3.00E+3nMAssay Description:Binding affinity to full length N-terminal His-tagged EED (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells by ITC methodMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataKd: 1.40E+4nMAssay Description:Binding affinity to G9a (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 97nMAssay Description:Binding affinity to Cbx4 (unknown origin) by ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+5nMAssay Description:Binding affinity to Cbx7 (unknown origin) by ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 5.00E+3nMAssay Description:Binding affinity to Cbx7 (unknown origin) by ITC methodMore data for this Ligand-Target Pair
Affinity DataKd: 850nMAssay Description:Binding affinity to C-terminal His-tagged CDYL2 (1 to 75 residues) (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells after 30 mins by fluor...More data for this Ligand-Target Pair
Affinity DataKd: 910nMAssay Description:Binding affinity to CDYL1b (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetTestis-specific chromodomain protein Y 1(Homo sapiens (Human))
University Of Connecticut
Curated by ChEMBL
University Of Connecticut
Curated by ChEMBL
Affinity DataKd: 6.30E+3nMAssay Description:Binding affinity to N-terminal GST-tagged CDY1 (1 to 101 residues) (unknown origin) expressed in Rosetta2 BL21(DE3)pLysS cells after 30 mins by fluor...More data for this Ligand-Target Pair