Compile Data Set for Download or QSAR
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Found 11 Enz. Inhib. hit(s) with all data for entry = 50000533
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252823(CHEMBL4077815)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in HEK293T cells assessed as inhibition of estradiol-induced response after 24 hrs by lucif...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252839(CHEMBL4082196)
Affinity DataIC50:  112nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in HEK293T cells assessed as inhibition of estradiol-induced response after 24 hrs by lucif...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252867(CHEMBL4074046)
Affinity DataIC50:  219nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in HEK293T cells assessed as inhibition of estradiol-induced response after 24 hrs by lucif...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252836(CHEMBL2413896)
Affinity DataIC50:  222nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in HEK293T cells assessed as inhibition of estradiol-induced response after 24 hrs by lucif...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252822(CHEMBL4076313)
Affinity DataIC50:  1.24E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in HEK293T cells assessed as inhibition of estradiol-induced response after 24 hrs by lucif...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252836(CHEMBL2413896)
Affinity DataEC50:  12nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in HEK293T cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252840(CHEMBL4081898)
Affinity DataEC50:  343nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in HEK293T cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252822(CHEMBL4076313)
Affinity DataEC50:  894nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in HEK293T cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252838(CHEMBL4062467)
Affinity DataEC50:  207nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in HEK293T cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252837(CHEMBL1915315)
Affinity DataEC50:  542nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in HEK293T cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wuhan University School of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50252839(CHEMBL4082196)
Affinity DataEC50:  11nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in HEK293T cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed