Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50049005
TargetNT-3 growth factor receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50232773(CHEMBL4091670)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of human TrkC using poly[Glu:Tyr] (4:1) as substrate preincubated for 20 mins followed by [gamma33P]ATP addition measured after 2 hrs by H...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50232773(CHEMBL4091670)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of human c-Kit using poly[Glu:Tyr] (4:1) as substrate preincubated for 20 mins followed by [gamma33P]ATP addition measured after 2 hrs by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50232773(CHEMBL4091670)
Affinity DataIC50:  19nMAssay Description:Inhibition of human FLT3 using EAIYAAPFAKKK as substrate preincubated for 20 mins followed by [gamma33P]ATP addition measured after 2 hrs by Hotspot ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50232774(CHEMBL4061775)
Affinity DataIC50:  217nMAssay Description:Inhibition of human FLT3 using EAIYAAPFAKKK as substrate preincubated for 20 mins followed by [gamma33P]ATP addition measured after 2 hrs by Hotspot ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50232775(CHEMBL4078141)
Affinity DataIC50:  359nMAssay Description:Inhibition of human FLT3 using EAIYAAPFAKKK as substrate preincubated for 20 mins followed by [gamma33P]ATP addition measured after 2 hrs by Hotspot ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed