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Found 12 Enz. Inhib. hit(s) with all data for entry = 50000844
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261657(CHEMBL4075572)
Affinity DataKd:  6.30nMAssay Description:Inhibition of p53 binding to MDM2 (unknown origin) after 30 mins by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261654(CHEMBL4076935)
Affinity DataKd:  15nMAssay Description:Inhibition of p53 binding to MDM2 (unknown origin) after 30 mins by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261655(CHEMBL4090785)
Affinity DataKd:  8.60nMAssay Description:Inhibition of p53 binding to MDM2 (unknown origin) after 30 mins by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261656(CHEMBL3347578)
Affinity DataKd:  3.20nMAssay Description:Inhibition of p53 binding to MDM2 (unknown origin) after 30 mins by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261655(CHEMBL4090785)
Affinity DataKd:  21nMAssay Description:Component deacylation rate constant for interaction with human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261658(CHEMBL4099164)
Affinity DataKd:  14nMAssay Description:Agonist activity at human beta-2 adrenergic receptor expressed in human H292 cells assessed as accumulation of intracellular cAMP after 1 hr by Alpha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261658(CHEMBL4099164)
Affinity DataKd:  61nMAssay Description:Cross Resistance (antiviral activity) of the compound with Y188C (Nonnucleoside reverse transcriptase inhibitor) resistant HIV isolate from cytopathi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261659(CHEMBL4059725)
Affinity DataKd:  346nMAssay Description:Cross Resistance (antiviral activity) of the compound with L100I (Nonnucleoside reverse transcriptase inhibitor) resistant HIV isolatefrom cytopathic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261659(CHEMBL4059725)
Affinity DataKd:  614nMAssay Description:HIV Protease inhibitory activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261656(CHEMBL3347578)
Affinity DataKd:  8.5nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in mouse A9 cells assessed as inositol phosphate accumulation using [myo-3H]inositol after 1 hr ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261657(CHEMBL4075572)
Affinity DataKd:  19nMAssay Description:Agonist activity at human beta-2 adrenergic receptor expressed in human H292 cells assessed as accumulation of intracellular cAMP after 1 hr by Alpha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50261654(CHEMBL4076935)
Affinity DataKd:  84nMAssay Description:Binding affinity towards muscarinic acetylcholine receptor by inhibiting specific binding of [3H]-quinuclidinyl benzilate (0.8 nM) in vitro to membra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed