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Found 8 Enz. Inhib. hit(s) with all data for entry = 50001184
TargetSerine/threonine-protein kinase ULK2(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of GST-tagged ULK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of GST-tagged ULK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50:  8nMAssay Description:Inhibition of N-terminal SUMO-tagged ULK1 kinase domain (1 to 283 residues) (unknown origin) using MBP as substrate in presence of [32P]ATP after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK2(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50271370(CHEMBL4127042)
Affinity DataIC50:  38nMAssay Description:Inhibition of GST-tagged ULK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50271370(CHEMBL4127042)
Affinity DataIC50:  45nMAssay Description:Inhibition of GST-tagged ULK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM379177(2-(5-Bromo-2-(3,4,5-trimethoxyphenylamino)pyrimidi...)
Affinity DataIC50:  108nMAssay Description:Inhibition of GST-tagged ULK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK2(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM379177(2-(5-Bromo-2-(3,4,5-trimethoxyphenylamino)pyrimidi...)
Affinity DataIC50:  711nMAssay Description:Inhibition of GST-tagged ULK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
Sichuan Universitt China Hospital

Curated by ChEMBL
LigandPNGBDBM50271371(CHEMBL4125718)
Affinity DataEC50:  19nMAssay Description:Activation of recombinant human N-terminal GST-tagged ULK1 (1 to 649 residues) expressed in baculovirus infected Sf9 cells using MBP as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed