Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50003190
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50468000(CHEMBL4288251)
Affinity DataEC50:  400nMAssay Description:Agonist activity at recombinant full length human LRH1 expressed in HeLa cells after 24 hrs by dual-glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50418303(CHEMBL1765959)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at recombinant full length human LRH1 expressed in HeLa cells after 24 hrs by dual-glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50467999(CHEMBL4291058)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at recombinant full length human LRH1 expressed in HeLa cells after 24 hrs by dual-glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50467997(CHEMBL4277194)
Affinity DataEC50:  1.30E+4nMAssay Description:Agonist activity at recombinant full length human LRH1 expressed in HeLa cells after 24 hrs by dual-glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50467998(CHEMBL4288877)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at recombinant full length human LRH1 expressed in HeLa cells after 24 hrs by dual-glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed