Compile Data Set for Download or QSAR
Report error Found 1 Enz. Inhib. hit(s) with all data for entry = 50004998
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Ponce De Leon Health

Curated by ChEMBL
LigandPNGBDBM50378137(Ketek | TELITHROMYCIN)
Affinity DataEC50:  1.32E+5nMAssay Description:Inhibition of human alpha3beta4 nAChR assessed as increase in acetylcholine-induced normalized current at 2 uM (Rvb = 78.5 +/- 10 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed