Found 14 Enz. Inhib. hit(s) with all data for entry = 50011295 
Affinity DataKi: 14nMAssay Description:Inhibition of recombinant human MMP2 expressed in human HeLaS3 cells using MOCAcPLGLA2pr(Dnp)-AR-NH2 as substrate incubated for 15 to 30 mins by fluo...More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibition of recombinant human MMP9 expressed in human HeLaS3 cells using MOCAcPLGLA2pr(Dnp)-AR-NH2 as substrate incubated for 15 to 30 mins by fluo...More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of recombinant human MMP12 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 30nMAssay Description:Inhibition of MMP2 (unknown origin) using 3163v as substrate preincubated for 15 mins followed by substrate addition and measured after 40 mins by fl...More data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of human MMP9 measured at 5 mins interval for 1 hr by fluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of human proMMP9 expressed in African green monkey COS-1 cells assessed as reduction in protein activation incubated for 30 mins prior to ...More data for this Ligand-Target Pair
Affinity DataIC50: 656nMAssay Description:Inhibition of human MMP2 measured at 5 mins interval for 1 hr by fluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human MT1-MMP using 3163v as substrate preincubated for 15 mins followed by substrate addition and measured after 40 mins by fluorometr...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human MMP9 using 3163v as substrate preincubated for 15 mins followed by substrate addition and measured after 40 mins by fluorometric ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MMP3 (unknown origin) using 3168v as substrate preincubated for 15 mins followed by substrate addition and measured after 40 mins by fl...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human MMP7 using 3163v as substrate preincubated for 15 mins followed by substrate addition and measured after 40 mins by fluorometric ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MT1-MMP catalytic domain (unknown origin) expressed in Escherichia coli using 7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-[2,4-din...More data for this Ligand-Target Pair
Affinity DataKd: 320nMAssay Description:Binding affinity to C-terminal 8-His tagged human MMP-9 hemopexin-like domain (Ala20 to Asp707 residues) expressed in 293E cells by fluorescence spec...More data for this Ligand-Target Pair
Affinity DataKd: 2.10E+3nMAssay Description:Binding affinity to MMP9 (unknown origin) by fluorescence spectroscopyMore data for this Ligand-Target Pair
