Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.10nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 57nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 61nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 81nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 283nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 34nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 68nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 68nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as IL-17 production by ELISAMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Bristol Myers Squibb
Curated by ChEMBL
Bristol Myers Squibb
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Inverse agonist activity at PXR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: >7.50E+3nMAssay Description:Inverse agonist activity at LXRbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at Gal4-fused RORalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 8.40E+3nMAssay Description:Inverse agonist activity at Gal4-fused RORbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Inverse agonist activity at RORgammat in mouse Th17 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >7.50E+3nMAssay Description:Inverse agonist activity at LXRalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 26nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.5nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair