Compile Data Set for Download or QSAR
maximum 50k data
Found 75 Enz. Inhib. hit(s) with all data for entry = 50013143
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50257829(2-(4-amino-5-(5-iodo-2-isopropyl-4-methoxyphenoxy)...)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183138(US9150546, I-291 | US9688643, I-291 | US9718790, I...)
Affinity DataIC50:  9.10nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183166(US9150546, I-326 | US9688643, I-326 | US9718790, I...)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183191(US9150546, I-355 | US9688643, I-355 | US9718790, I...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183184(US9150546, I-348 | US9688643, I-348 | US9718790, I...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183132(US9150546, I-285 | US9688643, I-285 | US9718790, I...)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563052(CHEMBL4748113)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183201(US9150546, I-365 | US9688643, I-365 | US9718790, I...)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183266(US9150546, I-434 | US9688643, I-434 | US9718790, I...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183145(US9150546, I-298 | US9688643, I-298 | US9718790, I...)
Affinity DataIC50:  27nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183200(US9150546, I-364 | US9688643, I-364 | US9718790, I...)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183097(US9150546, I-228 | US9688643, I-228 | US9718790, I...)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183139(US9150546, I-292 | US9688643, I-292 | US9718790, I...)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563048(CHEMBL4789094)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183121(US9150546, I-273 | US9688643, I-273 | US9718790, I...)
Affinity DataIC50:  38nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183125(US9150546, I-277 | US9688643, I-277 | US9718790, I...)
Affinity DataIC50:  38nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183107(US9150546, I-244 | US9688643, I-244 | US9718790, I...)
Affinity DataIC50:  45nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2/3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50257829(2-(4-amino-5-(5-iodo-2-isopropyl-4-methoxyphenoxy)...)
Affinity DataIC50:  45nMAssay Description:Antagonist activity at human P2X2/3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183146(US9150546, I-299 | US9688643, I-299 | US9718790, I...)
Affinity DataIC50:  46nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183148(US9150546, I-301 | US9688643, I-301 | US9718790, I...)
Affinity DataIC50:  48nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183136(US9150546, I-289 | US9688643, I-289 | US9718790, I...)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183199(US9150546, I-363 | US9688643, I-363 | US9718790, I...)
Affinity DataIC50:  78nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183160(US9150546, I-320 | US9688643, I-320 | US9718790, I...)
Affinity DataIC50:  83nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183135(US9150546, I-288 | US9688643, I-288 | US9718790, I...)
Affinity DataIC50:  93nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183089(US9150546, I-200 | US9688643, I-200 | US9718790, I...)
Affinity DataIC50:  128nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50413382(CHEMBL494833)
Affinity DataIC50:  136nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563041(CHEMBL4746334)
Affinity DataIC50:  144nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563036(CHEMBL4787960)
Affinity DataIC50:  149nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563049(CHEMBL4752152)
Affinity DataIC50:  152nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183143(US9150546, I-296 | US9688643, I-296 | US9718790, I...)
Affinity DataIC50:  176nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563050(CHEMBL4796811)
Affinity DataIC50:  219nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183070(US9150546, I-020 | US9688643, I-020 | US9718790, I...)
Affinity DataIC50:  389nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183117(US9150546, I-269 | US9688643, I-269 | US9718790, I...)
Affinity DataIC50:  415nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183110(US9150546, I-248 | US9688643, I-248 | US9718790, I...)
Affinity DataIC50:  420nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183106(US9150546, I-243 | US9688643, I-243 | US9718790, I...)
Affinity DataIC50:  450nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183112(US9150546, I-255 | US9688643, I-255 | US9718790, I...)
Affinity DataIC50:  520nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563051(CHEMBL4788581)
Affinity DataIC50:  614nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183131(US9150546, I-284 | US9688643, I-284 | US9718790, I...)
Affinity DataIC50:  629nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183103(US9150546, I-240 | US9688643, I-240)
Affinity DataIC50:  953nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563037(CHEMBL4797969)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563035(CHEMBL4778429)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563053(CHEMBL4749540)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2/3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183200(US9150546, I-364 | US9688643, I-364 | US9718790, I...)
Affinity DataIC50:  2.37E+3nMAssay Description:Antagonist activity at human P2X2/3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2/3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563052(CHEMBL4748113)
Affinity DataIC50:  2.93E+3nMAssay Description:Antagonist activity at human P2X2/3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563045(CHEMBL4797152)
Affinity DataIC50: >3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563044(CHEMBL4743578)
Affinity DataIC50: >3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563043(CHEMBL4759101)
Affinity DataIC50: >3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563047(CHEMBL4750833)
Affinity DataIC50: >3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563040(CHEMBL4757743)
Affinity DataIC50: >3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563039(CHEMBL4746738)
Affinity DataIC50: >3.00E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in rat C6-BU-1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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