TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 5.90E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 7.70E+3nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 7.90E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 9.80E+3nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.11E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.13E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.21E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.32E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.36E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.55E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.84E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.88E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.17E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.29E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.53E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.94E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.96E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 3.06E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 3.97E+4nMAssay Description:Binding affinity to recombinant human N-terminal MBP tagged/C-terminal His-tagged human PLK3-PBD (335 to 646 residue) expressed in Escherichia coli e...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 9.83E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 1.18E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.24E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.59E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: >6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: >6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: >6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: >6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: >6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: >6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataIC50: >6.00E+5nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged PLK1-PBD (367 to 603 end residue) expressed in Escherichia coli using MAGPMQS[pT]PLNGAKK ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataEC50: 820nMAssay Description:Binding affinity to full length PLK1 in human PC-3 cells assessed as stabilized protein incubated for 2 hrs followed by aggregation temperature at 56...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
University Of South Carolina
Curated by ChEMBL
University Of South Carolina
Curated by ChEMBL
Affinity DataEC50: 6.90E+3nMAssay Description:Binding affinity to full length PLK3 in human PC-3 cells assessed as stabilized protein incubated for 2 hrs followed by aggregation temperature at 48...More data for this Ligand-Target Pair